As publicações listadas adiante são alguns exemplos representativos de trabalhos desenvolvidos no LQFar ou que são provenientes de participação de seus membros, como colaboradores, em projetos de outros grupos. Para conhecê-las na íntegra, é só seguir o link.
- 4-nitrobenzoylcoumarin potentiates the antiparasitic, anti-inflammatory and cardioprotective effects of benznidazole in a murine model of acute Trypanosoma cruzi infection.
- A New 1,2-Benzisoxazolin-3-one Synthetized from Eugenol Shows Anti- Candida Spp. Activity, Specially Against Opportunistic Candida Glabrata.
- Action of N-Succinyl and N,O-Dicarboxymethyl Chitosan Derivatives on Chlorophyll Photosynthesis and Fluorescence in Drought-Sensitive Maize.
- Allelochemical Activity of Eugenol-Derived Coumarins on Lactuca sativa L.
- Antifungal Activity of a Library of Aminothioxanthones.
- Antifungal Activity of New Eugenol-Benzoxazole Hybrids against Candida spp.
- Benzophenone Derivatives Showed Dual Anti-Inflammatory and Antiproliferative Activities by Inhibiting COX Enzymes and Promote Cyclin E Downregulation.
- Characterization of antimicrobial and antioxidant performance of dihydroeugenol and its glycoside incorporated into whey protein isolate films.
- Combining eugenol and dihydroeugenol with a piperazine moiety to create new antimicrobial agents that are effective against resistant species.
- Coumarins as Potential Antiprotozoal Agents: Biological Activities and Mechanism of Action.
- Design, Synthesis and Pharmacological Evaluation of Novel Antiinflammatory and Analgesic O-Benzyloxime Compounds Derived From Natural Eugenol.
- Design, Synthesis, Antimicrobial Evaluation and Studies of Eugenol-Sulfonamide Hybrids.
- Design, Synthesis, Biological Evaluation and Molecular Modeling Studies of Novel Eugenol Esters as Leishmanicidal Agents.
- Dihydroeugenol derivatives associated with blue LED light: A different form to face multidrug resistant (MDR) bacteria.
- Do chitosan and its derivatives have the same protective effect on drought-contrasting maize genotypes? An analysis of physiological and production processes.
- Evaluation of antiplasmodial activity in silico and in vitro of N-acylhydrazone derivatives.
- Exploring how structural changes to new Licarin A derivatives effects their bioactive properties against rapid growing mycobacteria and biofilm formation.
- From Antibacterial to Antitumour Agents: A Brief Review on The Chemical and Medicinal Aspects of Sulfonamides.
- Glucosyl-1,2,3-triazoles derived from eugenol and analogues: Synthesis, anti- Candida activity, and molecular modeling studies in CYP-51.
- In silico evaluation and in vitro growth inhibition of Plasmodium falciparum by natural amides and synthetic analogs.
- In vitro and in silico antibacterial evaluation of coumarin derivatives against MDR strains of Staphylococcus aureus and Escherichia coli.
- In vitro and in silico evaluation of the schistosomicidal activity of eugenol derivatives using biochemical, molecular, and morphological tools.
- In vitro and in vivo trypanocidal activities of 8-methoxy-3-(4-nitrobenzoyl)-6-propyl-2 -cromen-2-one, a new synthetic coumarin of low cytotoxicity against mammalian cells.
- Investigation of 8-methoxy-3-(4-nitrobenzoyl)-6-propyl-2H-chromen-2-one as a promising coumarin compound for the development of a new and orally effective antileishmanial agent.
- Leaf application of chitosan and physiological evaluation of maize hybrids contrasting for drought tolerance under water restriction.
- Molecular docking, quorum quenching effect, antibiofilm activity and safety profile of silver-complexed sulfonamide on.
- Natural and Semi-synthetic Licarins: Neolignans with Multi-functional Biological Properties.
- New Antifungal Agents with Azole Moieties.
- New eugenol glucoside-based derivative shows fungistatic and fungicidal activity against opportunistic Candida glabrata.
- New miconazole-based azoles derived from eugenol show activity against Candida spp. and Cryptococcus gattii by inhibiting the fungal ergosterol biosynthesis.
- Phenylpropanoid-based sulfonamide promotes cyclin D1 and cyclin E down-regulation and induces cell cycle arrest at G1/S transition in estrogen positive MCF-7 cell line.
- Photobiological effect of eugenol-derived 3-benzoylcoumarin associated with led lights against MDR microorganisms.
- Physicochemical characterization of chitosan and its effects on early growth, cell cycle and root anatomy of transgenic and non-transgenic maize hybrids.
- Relevance of Trypanothione Reductase Inhibitors on Trypanosoma cruzi Infection: A Systematic Review, Meta-Analysis, and In Silico Integrated Approach.
- Síntese e avaliação preliminar da atividade antibacteriana e antifúngica de derivados N-acilidrazônicos.
- Structure-based discovery of thiosemicarbazones as SARS-CoV-2 main protease inhibitors.
- Synthesis and antimicrobial activity of molecular hybrids based on eugenol and chloramphenicol pharmacophores.
- Synthesis and antimicrobial activity of 6-triazolo-6-deoxy eugenol glucosides.
- Synthesis and biological evaluation of new eugenol Mannich bases as promising antifungal agents.
- Synthesis and Biological Evaluation of New Eugenol-Derived 1,2,3-Triazoles as Antimycobacterial Agents.
- Synthesis and biological evaluation of novel piperidine-benzodioxole derivatives designed as potential leishmanicidal drug candidates.
- Synthesis and evaluation of marine-inspired compounds result in hybrids with antitrypanosomal and antileishmanial activities.
- Synthesis and in vitro evaluation of antifungal and cytotoxic activities of eugenol glycosides.
- Synthesis and in vitro evaluation of leishmanicidal activity of 7-hydroxy-4-phenylcoumarin derivatives.
- Synthesis and in vitro evaluation of peracetyl and deacetyl glycosides of eugenol, isoeugenol and dihydroeugenol acting against food-contaminating bacteria.
- Synthesis and structural characterization of new benzylidene glycosides, cytotoxicity against cancer cell lines and molecular modeling studies.
- Synthesis and Structure-Activity Relationship Studies of Novel Aryl Sulfonamides and Their Activity against Human Breast Cancer Cell Lines.
- Synthesis of eugenol-derived glucosides and evaluation of their ability in inhibiting the angiotensin converting enzyme.
- Synthesis of New Hybrid Derivatives from Metronidazole and Eugenol Analogues as Trypanocidal Agents.
- Synthesis of piplartine analogs and preliminary findings on structure-antimicrobial activity relationship.
- Synthesis, activity, and docking studies of eugenol-based glucosides as new agents against Candida sp.
- Synthesis, activity, and molecular modeling studies of 1,2,3-triazole derivatives from natural phenylpropanoids as new trypanocidal agents.
- Synthesis, chemical characterization and antimicrobial activity of new acylhydrazones derived from carbohydrates.
- Synthesis, protease inhibition, and antileishmanial activity of new benzoxazoles derived from acetophenone or benzophenone and synthetic precursors.
- Tagitinin F has anti-inflammatory, anti-nociceptive and anti-matrix metalloproteinase properties: An in silico, in vitro and in vivo study.
- The foliar application of a mixture of semisynthetic chitosan derivatives induces tolerance to water deficit in maize, improving the antioxidant system and increasing photosynthesis and grain yield.
- The relationship between the antimicrobial activity of eugenol and the LPETG peptide structure and associated analysis for docking purposes.